Important Safety Information for 2-in-1 (Avanafil/Tadalafil)
Sexual Health

2-in-1 (Avanafil/Tadalafil)

Combination therapy providing both fast-acting (Avanafil) and long-lasting (Tadalafil) effects for comprehensive erectile dysfunction treatment.

What is the FDA-approved use of Avanafil/Tadalafil combination?

This combination contains two PDE5 inhibitors that work together:

  • Avanafil provides rapid onset of action (15-30 minutes) for spontaneous sexual activity.
  • Tadalafil provides extended duration of action (up to 36 hours) for flexibility in timing.
  • Combined therapy for men with severe erectile dysfunction who don't respond to single-agent therapy.

Limitations of Use:

  • This combination is not FDA-approved and is used off-label.
  • Not recommended for men with cardiovascular disease.
  • Not suitable for daily use due to increased side effect risk.

This combination should only be used under strict medical supervision with regular cardiovascular monitoring.

Who should not use Avanafil/Tadalafil combination?

Do not use this combination if:

  • You are taking nitrates, alpha-blockers, or guanylate cyclase stimulators.
  • You have severe cardiovascular disease, uncontrolled hypertension, or recent stroke/heart attack.
  • You have liver or kidney impairment.
  • You are taking CYP3A4 inhibitors (certain antibiotics, antifungals).
  • You have a history of priapism or bleeding disorders.

How should Avanafil/Tadalafil combination be administered?

Take no more than one tablet in a 48-hour period. This extended interval is necessary due to the combination's prolonged effects and increased risk profile.

Critical: Never exceed the recommended dose. The combination significantly increases the risk of dangerous side effects compared to single-agent therapy.

Side Effects Information

Common Side Effects

Dermatologic

  • Flushing (15% to 25%)

Neurologic

  • Headache (40% to 55%)
  • Dizziness (8% to 12%)

Gastrointestinal

  • Indigestion (10% to 18%)

Musculoskeletal

  • Back pain (15% to 20%)
  • Muscle pain (10% to 18%)

Respiratory

  • Nasal congestion (10% to 20%)

Ophthalmic

  • Visual disturbances (5% to 10%)

Serious Side Effects

Cardiovascular

  • Severe hypotension
  • Myocardial infarction
  • Stroke
  • Arrhythmias

Reproductive

  • Priapism (prolonged erection)

Ophthalmic

  • Sudden vision loss (NAION)

Otic

  • Sudden hearing loss

Contact Information

Reach out to our support team for any questions or assistance.

This is an off-label combination therapy. Please consult your healthcare provider for complete safety information.